Design and synthesis of novel tacrine–indole hybrids as potential multitarget-directed ligands for the treatment of Alzheimer's disease
BackBibliographic information
- Publication year
- 2021
- Category
- ADM — Scientific papers in foreign journals registered in Web of Science or SCOPUS databases
- CREPČ / EPCA ID
- 0037374
- Document type
- Journal article
- Source
- Future medicinal chemistry
- ISSN (Source)
- 1756-8919
- Volume
- Vol. 13, no. 9 (2021), p. 785-804
- Language
- English
- Research areas
- 200 — Veterinary Sciences
- Links
Bibliographic record
HAMUĽAKOVÁ, Slávka - KUDLIČKOVÁ, Zuzana - JANOVEC, Ladislav - MEZENCEV, Roman - DECKNER, Zachery J. - CHERNOFF, Yury O. - JANOČKOVÁ, Jana - IHNÁTOVÁ, Veronika - BZONEK, Petr - NOVÁKOVÁ, Nikola - HEPNÁROVÁ, Vendula - HRABINOVÁ, Martina - JUN, Daniel - KORÁBEČNÝ, Jan - SOUKUP, Ondrej - KUČA, Kamil. Design and synthesis of novel tacrine–indole hybrids as potential multitarget-directed ligands for the treatment of Alzheimer's disease. In: Future medicinal chemistry. 2021. ISSN 1756-8919, Vol. 13, no. 9 (2021), p. 785-804. (2021: 4.767 - IF, 76 - H-index, 4.791 - IF 5y, 0.649 - SJR, Q2 - SJR Best Q, Q2 - JCR Best Q, 0.809 - ABDC).
Publication authors
| Author | Role | Share |
|---|---|---|
| Slávka Hamuľaková | Author | 30.000 % |
| Zuzana Kudličková | Author | 10.000 % |
| Ladislav Janovec | Author | 10.000 % |
| Roman Mezencev | Author | 30.000 % |
| Zachery J. Deckner | Author | 5.000 % |
| Yury O. Chernoff | Author | 5.000 % |
| Jana Janočková | Author | 1.000 % |
| Veronika Ihnátová | Author | 1.000 % |
| Petr Bzonek | Author | 1.000 % |
| Nikola Nováková | Author | 1.000 % |
| Vendula Hepnárová | Author | 1.000 % |
| Martina Hrabinová | Author | 1.000 % |
| Daniel Jun | Author | 1.000 % |
| Jan Korábečný | Author | 1.000 % |
| Ondrej Soukup | Author | 1.000 % |
| Kamil Kuča | Author | 1.000 % |
Metrics
Citations (9)
| Citation year / Category | Citations | Source |
|---|---|---|
| 2025 1 |
DORABABU, Atukuri. Role of quinoline and indole-based heterocycles in revolutionizing Alzheimer's drug discovery: Promising futuristic structural designs. In JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 2025, vol. 392, no. 7, pp. ISSN 0022-3565. Dostupné na: https://doi.org/10.1016/j.jpet.2025.103606. |
WOS |
| 2025 1 |
SILVA SOUSA, Gleyton Leonel - NADUR, Nathalia Fonseca - DE ALMEIDA PEIXOTO FERREIRA, Larissa - DA SILVA HONÓRIO, Thiago - SIMON, Alice - CABRAL, Lucio Mendes - MÓRA SANTOS, Maria Luiza - ANDRADE, Bruna - DE LIMA, Emanuelle V. - CLARKE, Julia R. - CASTRO, Rosane Nora - OLÍMPIO DE MOURA, Ricardo - KÜMMERLE, Arthur Eugen. Discovery of novel thiosemicarbazone-acridine targeting butyrylcholinesterase with antioxidant, metal complexing and neuroprotector abilities as potential treatment of Alzheimer's disease: In vitro, in vivo, and in silico studies. In European Journal of Medicinal Chemistry, 2025-01-05, 281, pp. ISSN 02235234. Dostupné na: https://doi.org/10.1016/j.ejmech.2024.117030. |
WOS |
| 2024 1 |
IRAJI, Aida - NIKFAR, Parisa - NAZARI MONTAZER, Mohammad - KARIMI, Mona - EDRAKI, Najmeh - SAEEDI, Mina - MIRFAZLI, Seyedeh Sara. Synthesis, biological evaluation and molecular modeling studies of methyl indole-isoxazole carbohydrazide derivatives as multi-target anti-Alzheimer’s agents. In Scientific Reports, 2024-12-01, 14, 1, pp. Dostupné na: https://doi.org/10.1038/s41598-024-71729-0. |
SCOPUS |
| 2024 1 |
RAVINDAR, Lekkala - HASBULLAH, Siti Aishah - RAKESH, K. P. - RAHEEM, Saki - AGUSTAR, Hani Kartini - ISMAIL, Norzila - LING, Lau Yee - HASSAN, Nurul Izzaty. Exploring diverse frontiers: Advancements of bioactive 4-aminoquinoline-based molecular hybrids in targeted therapeutics and beyond. In European Journal of Medicinal Chemistry, 2024-01-15, 264, pp. ISSN 02235234. Dostupné na: https://doi.org/10.1016/j.ejmech.2023.116043. |
WOS |
| 2023 1 |
BELINSKAIA, Daria A. - VORONINA, Polina A. - KRIVOROTOV, Denis V. - JENKINS, Richard O. - GONCHAROV, Nikolay V. Anticholinesterase and Serotoninergic Evaluation of Benzimidazole–Carboxamides as Potential Multifunctional Agents for the Treatment of Alzheimer’s Disease. In Pharmaceutics, 2023-08-01, 15, 8, pp. Dostupné na: https://doi.org/10.3390/pharmaceutics15082159. |
SCOPUS |
| 2023 1 |
CHELUSNOVA, Yu V. - VORONINA, P. A. - BELINSKAIA, D. A. - GONCHAROV, N. V. Benzimidazole-Carboxamides as Potential Therapeutics for Alzheimer’s Disease: Primary Analysis In Silico and In Vitro. In Bulletin of Experimental Biology and Medicine, 2023-07-01, 175, 3, pp. 345-352. ISSN 00074888. Dostupné na: https://doi.org/10.1007/s10517-023-05865-4. |
SCOPUS |
| 2023 1 |
LI, Zhao Hui - YIN, Li Quan - ZHAO, Dong Hai - JIN, Lian Hai - SUN, Ya Juan - TAN, Cheng. SAR studies of quinoline and derivatives as potential treatments for Alzheimer's disease. In Arabian Journal of Chemistry, 2023-02-01, 16, 2, pp. ISSN 18785352. Dostupné na: https://doi.org/10.1016/j.arabjc.2022.104502. |
SCOPUS |
| 2023 1 |
PANADA, Jan - KLOPAVA, Valeriya - KULAHAVA, Tatsiana - KORAN, Siarhei - FALETROV, Yaroslav - FROLOVA, Nina - FOMINA, Elena - SHKUMATOV, Vladimir. Differential induction of C6 glioma apoptosis and autophagy by 3β-hydroxysteroid-indolamine conjugates. In Steroids, 2023-12-01, 200, pp. ISSN 0039128X. Dostupné na: https://doi.org/10.1016/j.steroids.2023.109326. |
SCOPUS |
| 2022 1 |
ZHANG, Honghua - PENG, Yan - ZHUO, Linsheng - WANG, Yuying - ZENG, Guo - WANG, Shuzhi - LONG, Lin - LI, Xuelin - WANG, Zhen. Recent advance on pleiotropic cholinesterase inhibitors bearing amyloid modulation efficacy. In EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, vol. 242, no., pp. ISSN 0223-5234. Dostupné na: https://doi.org/10.1016/j.ejmech.2022.114695. |
WOS |